SCHEMBL8050339

SCHEMBL8050339

COc1ccc2sc(-c3ccccn3)nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.60
SMN1; SMN2 Q16637 4/20 0.60
NPC1 O15118 4/20 0.60
KDM4E B2RXH2 3/20 0.60
ALDH1A1 P00352 2/20 0.60
TP53 P04637 1/20 0.60
TSHR P16473 1/20 0.60
HSD17B10 Q99714 1/20 0.60
DYRK1A Q13627 9/20 0.53
PKM P14618 1/20 0.51
TDP1 Q9NUW8 2/20 0.51
MAPT P10636 1/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
RUNX1 Q01196 1/20 0.51
MEN1 O00255 1/20 0.50
HPGD P15428 1/20 0.50
KMT2A Q03164 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11782932 0.90 RAB9A (0.63) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL23954341 0.81 KDM4E (0.77) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL8359494 0.81 KDM4E (0.50) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL2954313 0.80 MIF (0.65) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL20068807 0.79 SMN1; SMN2 (0.50) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL11780136 0.79 KDM4E (0.55) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL8054624 0.78 ALDH1A1 (0.51) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL8040079 0.78 KDM4E (0.66) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL29081219 0.78 KDM4E (0.66) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL3207351 0.78 NPC1 (0.66) RAB9ASMN1; SMN2NPC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed