SCHEMBL8041282

SCHEMBL8041282

COc1ccc(CCn2c3c(c4cc(C(C)N5CCc6c(c7cc(C)ccc7n6CCc6ccc(OC)cc6)C5)ccc42)CN(C)CC3)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.81
HRH1 P35367 16/20 0.81
ADRA2A P08913 3/20 0.67
HTR2A P28223 3/20 0.67
HTR2C P28335 3/20 0.67
HTR7 P34969 3/20 0.67
ADRA1A P35348 3/20 0.67
DRD2 P14416 2/20 0.62
GRIN1 Q05586 2/20 0.58
GRIN2A Q12879 2/20 0.58
GRIN2B Q13224 2/20 0.58
BCHE P06276 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
ACHE P22303 1/20 0.58
HRH2 P25021 1/20 0.58
ADRA1D P25100 1/20 0.58
HTR1D P28221 1/20 0.58
HTR1E P28566 1/20 0.58
ADRA1B P35368 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8036359 0.93 HTR6 (0.70) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL8031143 0.90 HTR6 (1.00) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL8036730 0.89 HTR6 (0.80) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL8044408 0.88 HTR6 (0.67) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL8034682 0.84 HTR6 (0.88) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL8032473 0.84 HTR6 (0.88) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL12881949 0.84 HTR6 (0.83) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL13696256 0.83 HTR6 (0.79) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL3715259 0.82 HTR6 (1.00) HTR6HRH1ADRA2AHTR2AHTR2C
SCHEMBL4140538 0.80 HTR6 (0.81) HTR6HRH1ADRA2AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009082268-A2 LIGANDS OF α-ADRENOCEPTORS AND OF DOPAMINE, HISTAMINE, IMIDAZOLINE AND SEROTONIN RECEPTORS AND THE USE THEREOF ALLA CHEM, LLC (US) 2009-07-02 WO disclosed