SCHEMBL8041296

SCHEMBL8041296

CCCCN(CCCN1CCOCC1)c1nc2c(CCC)nn(C)c2c(=O)[nH]1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 13/20 0.48
PDE6C P51160 1/20 0.46
MTOR P42345 1/20 0.41
TERT O14746 2/20 0.41
KMT2A Q03164 3/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4125332 0.86 PDE5A (0.46) PDE5APDE6CMTORTERTKMT2A
SCHEMBL4142307 0.85 PDE5A (0.47) PDE5APDE6CMTORTERTKMT2A
SCHEMBL8043292 0.85 PDE5A (0.45) PDE5APDE6CMTORTERTKMT2A
SCHEMBL8051166 0.85 PDE5A (0.45) PDE5APDE6CMTORTERTKMT2A
SCHEMBL8044800 0.83 PDE5A (0.44) PDE5APDE6CMTORTERTKMT2A
SCHEMBL4902005 0.81 PDE5A (0.56) PDE5APDE6CMTORTERTKMT2A
SCHEMBL4125201 0.78 PDE5A (0.36) PDE5APDE6CKMT2AHPGDALDH1A1
SCHEMBL4897792 0.75 PDE5A (0.46) PDE5APDE6CMTORTERTKMT2A
SCHEMBL4900871 0.74 PDE5A (0.48) PDE5APDE6CMTORKMT2AHPGD
SCHEMBL4136563 0.74 PDE5A (0.43) PDE5APDE6CMTORTERTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed