SCHEMBL8041300

SCHEMBL8041300

C=CC[C@H](CNCC)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.38
SLC6A4 P31645 14/20 0.38
SLC6A3 Q01959 14/20 0.38
CYP3A4 P08684 11/20 0.38
CYP2D6 P10635 11/20 0.38
KCNH2 Q12809 9/20 0.38
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6424063 0.85 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6424065 0.85 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL14144546 0.83 SMN1; SMN2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL13964798 0.82 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL13965179 0.80 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6604797 0.78 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6604805 0.78 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL4260062 0.77 SLC6A2 (0.33) SLC6A2SLC6A4ALDH1A1LMNA
SCHEMBL4027724 0.77 TBXAS1 (0.38) SLC6A2SLC6A4SLC6A3ALDH1A1LMNA
SCHEMBL6577169 0.76 SLC6A3 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136827-A PIPERIDINE COMPOUNDS AS DRUGS MERCK & CO., INC. (US) 2000-10-24 US disclosed
EP-1003514-A1 CYCLIC AMINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2000-05-31 EP disclosed
WO-1999004794-A1 CYCLIC AMINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1999-02-04 WO disclosed