SCHEMBL8041928

SCHEMBL8041928

O=C(O)/C(=C\c1ccccc1)CBr

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
AKR1C3 P42330 1/20 0.55
RECQL P46063 1/20 0.52
AKR1C1 Q04828 1/20 0.48
HTT P42858 1/20 0.46
MME P08473 2/20 0.45
PTPN1 P18031 1/20 0.43
GSK3B P49841 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TP53 P04637 1/20 0.42
FBP1 P09467 1/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
OPRK1 P41145 1/20 0.40
GRIK1 P39086 1/20 0.40
HAO1 Q9UJM8 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4327979 1.00 CYP3A4 (0.63) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL781849 1.00 CYP3A4 (0.63) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL8865069 0.89 TP53 (0.59) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL8865055 0.89 TP53 (0.59) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL8864851 0.84 CYP3A4 (0.47) CYP3A4CYP2C9AKR1C3HTTMEN1
SCHEMBL8864844 0.84 CYP3A4 (0.47) CYP3A4CYP2C9AKR1C3HTTMEN1
SCHEMBL2347233 0.84 CYP3A4 (0.50) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL8575022 0.84 CYP3A4 (0.59) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL7826083 0.84 CYP3A4 (0.47) CYP3A4CYP2C9AKR1C3RECQLAKR1C1
SCHEMBL7826086 0.84 CYP3A4 (0.47) CYP3A4CYP2C9AKR1C3RECQLAKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000024-A1 MERCAPTOACYLAMINO ACIDS AS METALLO-BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2000-05-17 EP disclosed
WO-1999006365-A1 MERCAPTOACYLAMINO ACIDS AS METALLO-BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-02-11 WO disclosed
US-5378711-A α-arylacrylates substituted by a heterocyclic radical, and fungicides which contain these compounds BASF AKTIENGESELLSCHAFT (DE) 1995-01-03 US disclosed
US-5326767-A α-arylacrylates substituted by a heterocyclic radical, and fungicides which contain these compounds BASF AKTIENGESELLSCHAFT (DE) 1994-07-05 US disclosed
US-5194438-A Plant safe fungicides BASF AKTIENGESELLSCHAFT (DE) 1993-03-16 US disclosed
US-5157037-A α-arylacrylates substituted by a heterocyclic radical, and fungicides which contain these compounds BASF AKTIENGESELLSCHAFT (DE) 1992-10-20 US disclosed