SCHEMBL8043092

SCHEMBL8043092

NC(=O)[C@H](CO)NCCCCOC1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.36
SPHK1 Q9NYA1 6/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPC1 O15118 1/20 0.32
BCHE P06276 1/20 0.32
F2 P00734 6/20 0.31
PRSS1 P07477 6/20 0.31
TERT O14746 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055986 0.96 NAAA (0.37) NAAAALDH1A1NPC1BCHEF2
SCHEMBL8055782 0.90 NPC1 (0.34) NAAANPC1F2PRSS1EPHX1
SCHEMBL971738 0.78 BCHE (0.44) BCHEEPHX1
SCHEMBL8043089 0.75 METAP2 (0.40) NAAASPHK1TERTEPHX1
SCHEMBL10431763 0.73 BCHE (0.44) BCHEEPHX1
SCHEMBL28417481 0.71 NAAA (0.42) NAAASPHK1KDM4EALDH1A1NPC1
SCHEMBL8055984 0.70 NAAA (0.40) NAAATERTEPHX1
SCHEMBL26203437 0.70 NPC1 (0.42) NAAASPHK1NPC1TERTEPHX1
SCHEMBL21842362 0.69 KDM4E (0.52) NAAAKDM4EEPHX1
SCHEMBL9011558 0.69 NPC1 (0.56) NAAASPHK1NPC1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114534-A REACTING A KETONE DERIVATIVE OF CARBAMOYL SUBSTITUTED HETEROCYCLE WITH PHOSPHORANE, FOLLOWED BY ACIDIFICATION TO FORM AN ANTICOAGULANT ELI LILLY AND COMPANY (US) 2000-09-05 US disclosed
US-6075147-A OMEGA-PHENYL-OMEGA-(3-PYRIDYL)-OMEGA-ALKENOIC ACID DERIVATIVES BEARING A CARBAMOYL SUBSTITUTED OXAZOLYL OR OXAZOLINYL GROUP ON THE PHENYL RING IS USEFUL FOR THROMBOXANE RECEPTOR ANTAGONSIM OR THROMBOXANE SYNTHASE INHIBITOR ELI LILLY AND COMPANY (US) 2000-06-13 US disclosed
US-6031095-A Intermediates in the preparation of substituted alkenoic acids ELI LILLY AND COMPANY (US) 2000-02-29 US disclosed
US-5990308-A Intermediates in the preparation of substituted alkenoic acids ELI LILLY AND COMPANY (US) 1999-11-23 US disclosed
US-5849922-A Preparation of substituted alkenoic acids ELI LILLY AND COMPANY (US) 1998-12-15 US disclosed
US-5849766-A Carbamoyl substituted heterocycles ELI LILLY AND COMPANY (US) 1998-12-15 US disclosed
EP-0816361-A2 Preparation of substituted alkenoic acids ELI LILLY AND COMPANY (US) 1998-01-07 EP disclosed
EP-0811621-A2 Carbamoyl substituted oxazoles as thromboxane receptor antagonists ELI LILLY AND COMPANY (US) 1997-12-10 EP disclosed