SCHEMBL8043146

SCHEMBL8043146

CC(C)(C)c1ccc(SCC(N)CO)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 1/20 0.44
KIF11 P52732 3/20 0.41
HRH3 Q9Y5N1 5/20 0.40
MAOA P21397 2/20 0.40
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MAOB P27338 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HRH4 Q9H3N8 3/20 0.38
CYP3A4 P08684 3/20 0.37
CYP2D6 P10635 3/20 0.37
CYP2C19 P33261 2/20 0.37
CYP1A2 P05177 2/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 2/20 0.36
TYR P14679 1/20 0.36
HSP90AA1 P07900 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17020095 0.77 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2MAOANPC1RAB9A
SCHEMBL3614462 0.76 MAOA (0.59) ALDH1A1KIF11MAOANPC1RAB9A
SCHEMBL3614466 0.76 MAOA (0.59) ALDH1A1KIF11MAOANPC1RAB9A
SCHEMBL27537594 0.75 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2HRH3NPC1RAB9A
Hydrochloric Acid SCHEMBL17009637 0.75 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2MAOANPC1RAB9A
SCHEMBL25005827 0.74 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2HRH3MAOANPC1
SCHEMBL12061831 0.74 TP53 (0.50) LMNATYR
SCHEMBL5231783 0.74 TP53 (0.50) LMNATYR
Ammonia Solution, Strong SCHEMBL7246795 0.74 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2HRH3MAOANPC1
SCHEMBL8031520 0.72 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2KIF11HRH3MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740659-B1 PHENYLTHIO-OXAZOLINE DERIVATIVES BAYER AG (DE) 2000-04-05 EP disclosed
CN-1138855-A Phenylthio-oxazoline derivatives BAYER AG (DE) 1996-12-25 CN disclosed
EP-0740659-A1 PHENYLTHIO-OXAZOLINE DERIVATIVES BAYER AG (DE) 1996-11-06 EP disclosed
WO-1995019348-A1 PHENYLTHIO-OXAZOLINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1995-07-20 WO disclosed