SCHEMBL8043339

SCHEMBL8043339

CCCCn1nnnc1Sc1ncc([N+](=O)[O-])s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
TLR9 Q9NR96 3/20 0.52
AGTR1 P30556 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPK8 P45983 7/20 0.49
MAPK9 P45984 7/20 0.49
MAPK10 P53779 2/20 0.45
ALDH1A1 P00352 5/20 0.43
HTT P42858 3/20 0.43
MAPT P10636 3/20 0.43
S1PR4 O95977 2/20 0.43
S1PR1 P21453 2/20 0.43
MAPK1 P28482 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
HSP90AA1 P07900 1/20 0.42
LMNA P02545 2/20 0.40
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046047 0.93 NPC1 (0.53) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8033453 0.88 NPC1 (0.58) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8032939 0.88 NPC1 (0.47) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8044040 0.88 MAPK8 (0.52) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8050061 0.85 NPC1 (0.45) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8050212 0.83 RAB9A (0.60) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8042307 0.82 MAPK8 (0.52) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8051088 0.81 NPC1 (0.45) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8032474 0.81 NPC1 (0.47) NPC1RAB9ATLR9AGTR1MEN1
SCHEMBL8046035 0.80 HTT (0.41) MEN1KMT2AALDH1A1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed