SCHEMBL8044575

SCHEMBL8044575

COc1nsc(NC(=O)N[C@@H](CC(C)C)C(=O)NCCC(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.41
CAPN9 O14815 2/20 0.41
ANPEP P15144 2/20 0.41
CTSB P07858 2/20 0.41
MAPK1 P28482 1/20 0.41
MMP3 P08254 1/20 0.40
CTSL P07711 2/20 0.40
LMNA P02545 1/20 0.40
CTSG P08311 1/20 0.40
FPR2 P25090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455524 0.84 ALDH1A1 (0.46) ANPEPMAPK1MMP3LMNAFPR2
SCHEMBL7642646 0.76 ANPEP (0.35) ANPEPMAPK1LMNA
SCHEMBL7406424 0.74 MEN1 (0.34) ANPEPLMNA
Proline SCHEMBL7402744 0.72 ALDH1A1 (0.36) MAPK1MMP3LMNAFPR2
SCHEMBL7442154 0.71 CYP2C9 (0.43)
SCHEMBL7402896 0.71 ALDH1A1 (0.36) MAPK1MMP3LMNAFPR2
Proline SCHEMBL7402894 0.71 SMN1; SMN2 (0.39) MMP3
SCHEMBL7397794 0.70 MEN1 (0.30) ANPEPLMNA
SCHEMBL22436168 0.68 ADORA3 (0.40)
SCHEMBL18941372 0.67 CAPN1 (0.62) CAPN1CAPN9ANPEPCTSBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed