SCHEMBL8044707

SCHEMBL8044707

O=C(O)c1sc(Sc2nnnn2-c2ccc(S(=O)(=O)Nc3ccccc3)cc2)nc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.43
NFE2L2 Q16236 2/20 0.43
EP300 Q09472 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.39
LIMK1 P53667 2/20 0.38
LIMK2 P53671 2/20 0.38
ALDH1A1 P00352 6/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043982 0.86 ALDH1A1 (0.47) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8051728 0.86 CA1 (0.44)
SCHEMBL8049019 0.82 RECQL (0.47) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8047493 0.82 CYP1A2 (0.40) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8048302 0.81 KMT2A (0.39) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8050392 0.81 EP300 (0.44) KEAP1NFE2L2EP300SMN1; SMN2LIMK1
SCHEMBL8042019 0.80 ALDH1A1 (0.39) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8048227 0.80 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL8046748 0.80 RECQL (0.39) EP300SMN1; SMN2ALDH1A1LMNATP53
SCHEMBL8044600 0.79 EP300 (0.46) KEAP1NFE2L2EP300SMN1; SMN2LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed