SCHEMBL8045596

SCHEMBL8045596

CN(C=O)CCCCCC/C=C/c1ccc2c(c1)/C(=N\O)c1ccccc1-2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.37
KDR P35968 4/20 0.37
AURKB Q96GD4 4/20 0.37
CDK5 Q00535 4/20 0.37
CDK5R1 Q15078 4/20 0.37
MAPT P10636 2/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HSP90AA1 P07900 2/20 0.33
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044206 1.00 AURKA (0.37) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8046738 0.79 HDAC1 (0.33) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8052434 0.79 HDAC1 (0.33) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8040097 0.77 KMT2A (0.47) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8045597 0.77 KMT2A (0.47) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8049240 0.76 AURKA (0.36) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8052442 0.74 AURKA (0.38) AURKAKDRAURKBCDK5CDK5R1
SCHEMBL8040840 0.67 POLB (0.34) HDAC1HDAC8MEN1KMT2A
SCHEMBL10352909 0.65 LMNA (0.32) MAPTHDAC1HDAC8HTTSMN1; SMN2
SCHEMBL8052878 0.65 POLB (0.35) HDAC1HDAC8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009085978-A1 BRIDGED CARBOCYCLIC OXIME HEPATITIS C VIRUS SERINE PROTEASE INHIBITORS ENANTA PHARCEUTICALS, INC. (US) 2009-07-09 WO disclosed