Pyrazine

Pyrazine

SCHEMBL8046266

N#Cc1nccnc1C#N.c1cnccn1.c1cncnc1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
PAX8 Q06710 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
GRM5 P41594 1/20 0.30
PLCG1 P19174 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrazine SCHEMBL27517504 0.88 ALDH1A1 (0.43) ALDH1A1LMNAMAPTPKMMAPK1
SCHEMBL217939 0.80 ALDH1A1 (0.38) ALDH1A1LMNAMAPTPKMMAPK1
SCHEMBL29350921 0.80 ALDH1A1 (0.38) ALDH1A1LMNAMAPTPKMMAPK1
Pyrazine SCHEMBL1428283 0.71 TSHR (0.54) ALDH1A1
Pyrimidine SCHEMBL1766109 0.67 TSHR (0.46) ALDH1A1
Pyrimidine SCHEMBL251837 0.67
Pyrimidine SCHEMBL28329992 0.67 TSHR (0.46) ALDH1A1
Pyrimidine SCHEMBL27488211 0.67
Pyrimidine SCHEMBL6978952 0.66
Pyrimidine SCHEMBL3502117 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991468-A1 HOMOGENEOUS OXIDATION CATALYSIS USING METAL COMPLEXES CARNEGIE-MELLON UNIVERSITY (US) 2000-04-12 EP disclosed
WO-1998058735-A1 HOMOGENEOUS OXIDATION CATALYSIS USING METAL COMPLEXES CARNEGIE MELLON UNIVERSITY (US) 1998-12-30 WO disclosed