SCHEMBL8046894

SCHEMBL8046894

CCCc1nc(SC)c(C(=O)OCC)n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.57
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP19A1 P11511 1/20 0.37
SIRT2 Q8IXJ6 2/20 0.36
SIRT1 Q96EB6 1/20 0.36
AGTR1 P30556 2/20 0.36
AGTR2 P50052 2/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HSD17B10 Q99714 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837125 0.88 EDNRA (0.70) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8432726 0.88 EDNRA (0.54) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8052641 0.87 EDNRA (0.54) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8045593 0.85 EDNRA (0.51) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8433056 0.85 EDNRA (0.53) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8049333 0.85 EDNRA (0.50) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8432727 0.84 EDNRA (0.58) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8044320 0.83 EDNRA (0.74) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8049397 0.83 EDNRA (0.49) EDNRAKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL8434967 0.83 EDNRA (0.63) EDNRAAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143774-A DRUGS AS HYPOTENSIVE AGENTS HOECHST MARION ROUSSEL (FR) 2000-11-07 US disclosed
US-5986103-A IMIDAZOLE SUBSTITUTED BENZENE AND REDUCTION OF ABNORMAL STIMULATION OF ENDOTHELIN RECEPTORS HOECHST MARION ROUSSEL (FR) 1999-11-16 US disclosed