SCHEMBL8047698

SCHEMBL8047698

O=C(c1ccc(OC/C=C/CBr)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.47
LSS P48449 3/20 0.47
MAOB P27338 3/20 0.47
PTPN1 P18031 1/20 0.46
GSK3B P49841 1/20 0.46
CYP1A1 P04798 2/20 0.45
CYP1B1 Q16678 2/20 0.45
ALDH1A1 P00352 1/20 0.43
GRM4 Q14833 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902485 1.00 SRD5A2 (0.47) SRD5A2LSSMAOBPTPN1GSK3B
SCHEMBL8902853 0.84 LSS (0.48) LSSMAOBPTPN1ALDH1A1
SCHEMBL8044759 0.84 LSS (0.48) LSSMAOBPTPN1ALDH1A1
SCHEMBL9360152 0.82 GAA (0.55) SRD5A2LSSALDH1A1
SCHEMBL9360157 0.82 GAA (0.55) SRD5A2LSSALDH1A1
SCHEMBL7685512 0.82 LSS (0.62) SRD5A2LSSMAOB
SCHEMBL7685521 0.82 LSS (0.62) SRD5A2LSSMAOB
SCHEMBL8903149 0.81 LSS (0.48) SRD5A2LSSALDH1A1
SCHEMBL8903155 0.81 LSS (0.48) SRD5A2LSSALDH1A1
SCHEMBL8905081 0.79 ALDH1A1 (0.49) LSSGSK3BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed