SCHEMBL8047723

SCHEMBL8047723

CCOC(=O)c1cc(-c2ccccc2)sc1NC(=O)NCCCl

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.69
HPGD P15428 7/20 0.69
LMNA P02545 2/20 0.69
KDM4E B2RXH2 3/20 0.66
TP53 P04637 1/20 0.66
THRB P10828 1/20 0.66
GSTO1 P78417 1/20 0.65
MAPT P10636 8/20 0.64
NPSR1 Q6W5P4 3/20 0.64
CNR2 P34972 1/20 0.61
GAA P10253 3/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2C19 P33261 2/20 0.60
HTT P42858 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.56
ALOX15 P16050 1/20 0.56
RAB9A P51151 1/20 0.56
HSD17B10 Q99714 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047722 0.83 HPGD (0.72) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL10732624 0.82 NPSR1 (0.50) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL5804319 0.80 ALDH1A1 (0.82) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL5804317 0.80 ALDH1A1 (0.82) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL4417698 0.79 ALDH1A1 (0.80) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL8051341 0.78 ALDH1A1 (0.64) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL1579548 0.78 ALDH1A1 (0.72) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL14875905 0.78 ALDH1A1 (0.76) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL3812791 0.78 ALDH1A1 (0.71) ALDH1A1HPGDLMNAKDM4ETP53
SCHEMBL5440410 0.77 HPGD (0.74) ALDH1A1HPGDLMNAKDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166019-A Piperazinyl pyrimidine dione compounds selective for adrenoceptors ABBOTT LABORATORIES (US) 2000-12-26 US disclosed
US-6153614-A Piperazinyl pyrimidine dione compounds selective for adrenoceptors ABBOTT LABORATORIES (US) 2000-11-28 US disclosed