SCHEMBL8048129

SCHEMBL8048129

Nc1ccc(-n2nnnc2S)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.38
NPSR1 Q6W5P4 3/20 0.38
HTT P42858 4/20 0.38
MAPT P10636 6/20 0.36
LMNA P02545 6/20 0.36
HPGD P15428 4/20 0.36
L3MBTL1 Q9Y468 4/20 0.36
HSP90AA1 P07900 2/20 0.36
CACNA1B Q00975 2/20 0.36
APBA1 Q02410 2/20 0.36
TP53 P04637 1/20 0.36
NLRP1 Q9C000 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
DHODH Q02127 1/20 0.36
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CCR6 P51684 1/20 0.34
TSHR P16473 3/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10011398 0.98 ALDH1A1 (0.37) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL8655762 0.89 ALDH1A1 (0.41) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL5685523 0.80 MAPT (0.56) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL14119061 0.80 ALDH1A1 (0.46) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL8048128 0.80 ALDH1A1 (0.49) ALDH1A1HTTMAPTLMNASMN1; SMN2
SCHEMBL594488 0.80 ALDH1A1 (0.47) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL6264097 0.80 ALDH1A1 (0.56) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL10022440 0.79 NOTUM (0.46) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL55213 0.79 ALDH1A1 (0.53) ALDH1A1NPSR1HTTMAPTLMNA
SCHEMBL27515853 0.78 ALDH1A1 (0.46) ALDH1A1NPSR1HTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1180310-C DIR compound and its application in preparing photosensitive material 中国乐凯胶片集团公司 2004-12-15 CN claimed
CN-1397837-A DIR compound and its application in preparing photosensitive material CHINESE LEKAI FILM GROUP CO (CN) 2003-02-19 CN claimed
US-6143765-A ENZYME IHIBITORS OF PROTEIN SUGEN, INC. (US) 2000-11-07 US disclosed
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
US-5883110-A ORGANIC MOLECULES CAPABLE OF INHIBITING PROTEIN TYROSINE PHOSPHATASE ACTIVITY, AND THE USE OF SUCH MOLECULES TO TREAT VARIOUS DISEASE STATES INCLUDING DIABETES MELLITUS, GLIOMA, MELANOMA, KAPOSI'S SARCOMA, HEMANGIOMA, OVARIAN CANCER, BREAST SUGEN, INC. (US) 1999-03-16 US disclosed
EP-0436027-B1 METHOD OF TREATING SILVER HALIDE PHOTOGRAPHIC MATERIAL FUJI PHOTO FILM CO LTD (JP) 1998-10-14 EP disclosed
US-5780198-A MULTILAYER; CONTAINS A HYDRAZINE NUCLEATING AGENT AND A REDOX COMPOUND CAPABLE OF RELEASING A DEVELOPMENT INHIBITOR WHEN THE REDOX COMPOUND IS OXIDIZED; ULTRAHIGH CONTRAST IMAGE WITH BROAD DOT GRADATION FUJI PHOTO FILM CO., LTD. (JP) 1998-07-14 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed
EP-0442323-B1 Silver halide color reversal photographic material capable of providing interimage effect FUJI PHOTO FILM CO LTD (JP) 1997-10-15 EP disclosed
EP-0218385-B2 Thermally developable light-sensitive material KONISHIROKU PHOTO IND (JP) 1997-05-14 EP disclosed
EP-0420005-B1 High contrast silver halide photographic material FUJI PHOTO FILM CO LTD (JP) 1996-07-10 EP disclosed
EP-0256820-A2 Thermal developing light-sensitive material KONICA CORPORATION (JP) 1988-02-24 EP disclosed
EP-0218385-A2 Thermally developable light-sensitive material KONICA CORPORATION (JP) 1987-04-15 EP disclosed
US-4554246-A THIOTETREAZOLYLPHENYL CARBAMATE FUJI PHOTO FILM CO., LTD. (JP) 1985-11-19 US disclosed
EP-0080631-B1 SILVER HALIDE PHOTOGRAPHIC LIGHT-SENSITIVE MATERIALS FUJI PHOTO FILM CO., LTD. (JP) 1985-06-26 EP disclosed
EP-0053851-B1 NOVEL ANTIFOGGING COMPOUNDS AND THEIR USE IN SILVER HALIDE PHOTOGRAPHY AGFA-GEVAERT N.V. (BE) 1985-05-29 EP disclosed
US-4451555-A 1-PHENYL-5-MERCAPTOTETRAZOLES AGFA-GEVAERT, N.V. (BE) 1984-05-29 US disclosed
US-4448878-A 1-(UREIDO-PHENYL), 5-MERCAPTO- 1H-TETRAZOLE COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1984-05-15 US disclosed
EP-0053851-A1 Novel antifogging compounds and their use in silver halide photography AGFA-GEVAERT N.V. (BE) 1982-06-16 EP disclosed
US-3708303-A PHOTOGRAPHIC ELEMENTS AND PROCESSES LITHOGRAPHIC SILVER HALIDE ELEMENT CONTAINING A 1-(AMIDOPHENYL)-5-MERCAPTOTETRAZOLE SENSITIZING AGENT AND DEVELOPMENT PROCESS OF USING SAME EASTMAN KODAK CO 1973-01-02 US disclosed