SCHEMBL8048680

SCHEMBL8048680

CSNC1CCN(CCC(C(=O)O)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 15/20 0.46
CCR5 P51681 2/20 0.45
TACR1 P25103 2/20 0.44
MCHR1 Q99705 2/20 0.42
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048710 0.90 SLC6A3 (0.50) TACR2TACR1SLC6A3
SCHEMBL295981 0.84 TACR2 (0.45) TACR2CCR5TACR1MCHR1
SCHEMBL10569422 0.77 GRIN2B (0.56) TACR2SLC6A3
SCHEMBL3637661 0.76 TACR2 (0.44) TACR2CCR5TACR1SLC6A3
SCHEMBL295129 0.74 SLC6A3 (0.49) TACR2CCR5TACR1SLC6A3
SCHEMBL8033015 0.74 KCNH2 (0.43) TACR2TACR1MCHR1
SCHEMBL295967 0.71 EPHX2 (0.43) TACR2CCR5TACR1MCHR1
SCHEMBL9734602 0.71 SLC6A3 (0.54) TACR2TACR1MCHR1SLC6A3
SCHEMBL297293 0.70 TACR3 (0.48) TACR2CCR5TACR1
SCHEMBL8095001 0.69 SLC6A3 (0.55) TACR2TACR1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033995-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-19 WO disclosed