SCHEMBL8049381

SCHEMBL8049381

C=CCN(c1ccncc1)c1csc2cc(Cl)ccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.33
CYP2A6 P11509 2/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
SLC6A2 P23975 2/20 0.31
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
DRD2 P14416 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
ADRA1D P25100 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR1E P28566 1/20 0.30
SLC6A4 P31645 1/20 0.30
HTR7 P34969 1/20 0.30
ADRA1A P35348 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8050441 0.99 ROCK1 (0.33) ROCK1CYP2A6NOS3NOS1NOS2
SCHEMBL8050457 0.86 ROCK1 (0.33) ROCK1CYP2A6MAPK1
Hydrochloric Acid SCHEMBL8053571 0.85 ROCK1 (0.33) ROCK1CYP2A6MAPK1
SCHEMBL8050470 0.85 ROCK1 (0.37) ROCK1CYP2A6NOS3NOS1NOS2
SCHEMBL8050534 0.84 ROCK1 (0.35) ROCK1CYP2A6NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL8051640 0.84 ROCK1 (0.36) ROCK1CYP2A6NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL8056254 0.83 ROCK1 (0.34) ROCK1CYP2A6NOS3NOS1NOS2
SCHEMBL8056707 0.82 SLC6A2 (0.41) ROCK1CYP2A6NOS3NOS1NOS2
SCHEMBL8049114 0.82 KIF11 (0.35)
Hydrochloric Acid SCHEMBL8038855 0.81 SLC6A2 (0.40) ROCK1CYP2A6NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022880-A Substituted pyridylamino indoles HOECHST MARION ROUSSEL, INC. (US) 2000-02-08 US disclosed
US-5328920-A Alleviating memory dysfunctions HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-07-12 US disclosed