SCHEMBL8049539

SCHEMBL8049539

CC(C)(C)OC(=O)N1C[C@H](NS(=O)(=O)c2cc(Cl)ccc2Cl)C[C@@H]1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.44
NR1H2 P55055 4/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
ALDH1A1 P00352 2/20 0.36
CPT2 P23786 1/20 0.36
CPT1A P50416 1/20 0.36
CPT1B Q92523 1/20 0.36
MAPT P10636 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
STS P08842 1/20 0.35
KDM4E B2RXH2 1/20 0.35
RORC P51449 1/20 0.34
F10 P00742 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047069 0.91 CPT2 (0.46) BRD4NR1H2CPT2CPT1ACPT1B
SCHEMBL3950906 0.88 ACLY (0.38) HSP90AA1HSP90AB1ALDH1A1CPT2CPT1A
SCHEMBL13663795 0.87 NR1H2 (0.37) BRD4NR1H2HSP90AA1HSP90AB1ALDH1A1
SCHEMBL8064460 0.84 NR1H2 (0.41) NR1H2HSP90AA1HSP90AB1ALDH1A1CPT2
SCHEMBL3954231 0.84 CTSL (0.46) BRD4NR1H2CTSLCTSBCTSS
SCHEMBL8063010 0.83 NR1H2 (0.41) BRD4NR1H2HSP90AA1HSP90AB1ALDH1A1
SCHEMBL8062643 0.83 CPT2 (0.45) NR1H2HSP90AA1HSP90AB1ALDH1A1CPT2
SCHEMBL8063921 0.82 CTSL (0.48) BRD4NR1H2ALDH1A1CTSLCTSB
SCHEMBL8063144 0.81 BRD4 (0.43) BRD4NR1H2ALDH1A1CPT2CPT1A
SCHEMBL13662001 0.81 F10 (0.36) BRD4HSP90AA1HSP90AB1ALDH1A1CPT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026197-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-02-26 WO disclosed