SCHEMBL8050280

SCHEMBL8050280

Oc1cccc(-c2csc(-c3ccccc3)n2)c1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.87
HSD17B2 P37059 1/20 0.87
CYP19A1 P11511 2/20 0.70
SMN1; SMN2 Q16637 5/20 0.69
KDM4E B2RXH2 4/20 0.69
KMT2A Q03164 4/20 0.69
MEN1 O00255 3/20 0.69
ALDH1A1 P00352 3/20 0.69
MAPT P10636 3/20 0.69
LMNA P02545 2/20 0.69
POLB P06746 2/20 0.69
GAA P10253 2/20 0.69
PKM P14618 2/20 0.69
HPGD P15428 2/20 0.69
ALOX12 P18054 2/20 0.69
SREBF2 Q12772 2/20 0.60
AR P10275 1/20 0.60
RAB9A P51151 3/20 0.59
CASP3 P42574 1/20 0.59
SENP8 Q96LD8 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180078 0.93 HSD17B1 (1.00) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL1181077 0.92 HSD17B1 (0.84) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL8057629 0.90 HSD17B1 (0.82) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL4267715 0.86 KDM4E (0.68) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL1180965 0.85 HSD17B1 (0.84) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL19195912 0.84 SMN1; SMN2 (0.66) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL8052755 0.83 HSD17B1 (0.75) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL8040175 0.83 CYP19A1 (0.74) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL6330424 0.83 SREBF2 (0.70) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E
SCHEMBL8051375 0.83 SREBF2 (0.70) HSD17B1HSD17B2CYP19A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed