SCHEMBL6330424

SCHEMBL6330424

Oc1ccc(-c2nc(-c3ccccc3)cs2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SREBF2 Q12772 1/20 0.70
CYP19A1 P11511 3/20 0.69
KDM4E B2RXH2 6/20 0.69
KMT2A Q03164 4/20 0.69
AR P10275 2/20 0.69
RAB9A P51151 6/20 0.69
SMN1; SMN2 Q16637 5/20 0.69
MAPT P10636 4/20 0.69
POLB P06746 3/20 0.69
MEN1 O00255 3/20 0.69
ALDH1A1 P00352 3/20 0.69
NPC1 O15118 3/20 0.69
LMNA P02545 2/20 0.69
GAA P10253 2/20 0.69
PKM P14618 2/20 0.69
HPGD P15428 2/20 0.69
ALOX12 P18054 2/20 0.69
ATM Q13315 1/20 0.67
USP2 O75604 1/20 0.66
HSP90AA1 P07900 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051375 1.00 SREBF2 (0.70) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL1181195 0.93 KDM4E (0.75) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL11212983 0.91 SREBF2 (0.82) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL11215130 0.91 SREBF2 (0.82) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL11213828 0.91 SREBF2 (0.82) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL11464717 0.89 SREBF2 (0.79) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL2781370 0.89 KDM4E (0.85) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL17409318 0.87 CYP19A1 (0.71) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL4267715 0.85 KDM4E (0.68) SREBF2CYP19A1KDM4EKMT2AAR
SCHEMBL1181077 0.85 HSD17B1 (0.84) SREBF2CYP19A1KDM4EKMT2AAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250270199-A1 THIAZOLE DERIVATIVES AND METHODS OF USING THE SAME ARKANSAS STATE UNIV JONESBORO (US) 2025-08-28 US claimed
US-20250270199-A1 THIAZOLE DERIVATIVES AND METHODS OF USING THE SAME ARKANSAS STATE UNIV JONESBORO (US) 2025-08-28 US disclosed
WO-2023192595-A1 THIAZOLE DERIVATIVES AND METHODS OF USING THE SAME Arkansas State University - Jonesboro (US) 2023-10-05 WO disclosed
US-20050075323-A1 Beta3 adrenergic receptor agonists and uses thereof PFIZER INC 2005-04-07 US disclosed
US-6706743-B2 β3 adrenergic receptor agonists and uses thereof PFIZER INC 2004-03-16 US disclosed
CN-1469876-A Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists �Ʒ� 2004-01-21 CN disclosed
US-20030203913-A1 Beta3 adrenergic receptor agonists and uses thereof PFIZER INC. 2003-10-30 US disclosed
EP-1326861-A1 ALPHA-ARYL ETHANOLAMINES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS Pfizer Products Inc. (US) 2003-07-16 EP disclosed
US-6566377-B2 β3 adrenergic receptor agonists and uses thereof PFIZER INC. 2003-05-20 US disclosed
US-20020052392-A1 Bita3 adrenergic receptor agonists and uses thereof DAY ROBERT F (US) 2002-05-02 US disclosed
WO-2002032897-A1 ALPHA-ARYL ETHANOLAMINES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS PFIZER PRODUCTS INC. (US) 2002-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030203913-A1 Beta3 adrenergic receptor agonists and uses thereof ADRB3, ADRB1, ADRB2 SREBF2 1434/4885CYP19A1 534/4885KDM4E 3213/4885
US-20050075323-A1 Beta3 adrenergic receptor agonists and uses thereof ADRB3, ADRB1, ADRB2 SREBF2 1734/4885CYP19A1 561/4885KDM4E 3070/4885
US-20250270199-A1 THIAZOLE DERIVATIVES AND METHODS OF USING THE SAME TST, GOT2, TPMT SREBF2 2545/4885CYP19A1 2098/4885KDM4E 4630/4885
US-20020052392-A1 Bita3 adrenergic receptor agonists and uses thereof ADRB3, ADRA1A, ADRB1 SREBF2 1970/4885CYP19A1 531/4885KDM4E 3754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.