SCHEMBL8050368

SCHEMBL8050368

BrCCOc1ccccc1-c1nc2ccccc2s1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
SMN1; SMN2 Q16637 6/20 0.52
NPC1 O15118 6/20 0.52
RAB9A P51151 6/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
KDM4E B2RXH2 6/20 0.51
MAPT P10636 6/20 0.51
GAA P10253 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
HCRTR1 O43613 1/20 0.49
GLA P06280 1/20 0.49
POLB P06746 1/20 0.47
HSD17B10 Q99714 3/20 0.45
TP53 P04637 2/20 0.45
TSHR P16473 1/20 0.45
HPGD P15428 2/20 0.45
PKM P14618 1/20 0.45
NPSR1 Q6W5P4 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24556005 0.91 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL25060427 0.82 KDM4E (0.60) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL25711522 0.81 NPC1 (0.51) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL25068629 0.80 KDM4E (0.62) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL21131752 0.77 KDM4E (0.63) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL21753766 0.77 NPC1 (0.58) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL23465937 0.77 NPC1 (0.58) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL20959856 0.77 NPC1 (0.58) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL21752785 0.77 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2088155 0.77 NPC1 (0.58) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed