SCHEMBL8051689

SCHEMBL8051689

CN(c1ccncc1)c1csc2ccc(C(F)(F)F)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 1/20 0.40
RIPK2 O43353 1/20 0.40
STK16 O75716 1/20 0.40
EGFR P00533 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
BMP2K Q9NSY1 1/20 0.40
NLK Q9UBE8 1/20 0.40
IRAK3 Q9Y616 1/20 0.40
POLQ O75417 1/20 0.39
KIF11 P52732 3/20 0.39
CHUK O15111 1/20 0.35
KDM4C Q9H3R0 2/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
GPBAR1 Q8TDU6 3/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8050875 0.99 GAK (0.39) GAKRIPK2STK16EGFRAAK1
SCHEMBL8052621 0.90 POLQ (0.39) GAKRIPK2STK16EGFRAAK1
Hydrochloric Acid SCHEMBL8038783 0.88 POLQ (0.39) GAKRIPK2STK16EGFRAAK1
SCHEMBL8056490 0.82 POLQ (0.36) GAKRIPK2STK16EGFRAAK1
SCHEMBL8038898 0.81 POLQ (0.35) AAK1POLQKIF11CHUKPIM1
Hydrochloric Acid SCHEMBL8050511 0.81 POLQ (0.35) POLQKIF11CHUKPIM1PIM2
Hydrochloric Acid SCHEMBL8049583 0.80 POLQ (0.35) POLQKIF11CHUKPIM1PIM2
SCHEMBL8039461 0.76 MAPT (0.39) MAPTMAPK1CHRM5CHKA
SCHEMBL8440409 0.76 CYP2A6 (0.43) MAPTCHRM5CHKA
Hydrochloric Acid SCHEMBL8039050 0.75 MAPT (0.38) MAPTMAPK1CHRM5CHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022880-A Substituted pyridylamino indoles HOECHST MARION ROUSSEL, INC. (US) 2000-02-08 US disclosed
US-5328920-A Alleviating memory dysfunctions HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-07-12 US disclosed