SCHEMBL8051960

SCHEMBL8051960

[CH]=CCc1ccoc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262869 0.78
SCHEMBL1994157 0.76
SCHEMBL16992903 0.73
SCHEMBL8670493 0.73 HCAR2 (0.38)
SCHEMBL9851139 0.72
SCHEMBL2840244 0.72
SCHEMBL14877408 0.71
SCHEMBL8670495 0.71 ALOX5 (0.43)
SCHEMBL8806436 0.69 ALOX5 (0.36)
SCHEMBL8198507 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2670406-B1 COMBINATION THERAPY WITH INTERFERON BETA AND ANDROGRAPHOLIDES FOR MULTIPLE SCLEROSIS INNOBIOSCIENCE LLC (US) 2015-09-02 EP claimed
US-9060994-B2 Combination therapy with interferon and andrographolides for Multiple Sclerosis Inno Biosciences, S.p.A. (CL) 2015-06-23 US claimed
US-20140301981-A1 Combination Therapy with Interferon and Andrographolides for Multiple Sclerosis INNOBIOSCIENCE LLC (US) 2014-10-09 US claimed
EP-2670406-A1 COMBINATION THERAPY WITH INTERFERON AND ANDROGRAPHOLIDES FOR MULTIPLE SCLEROSIS Herbal Powers Corporation (US) 2013-12-11 EP claimed
WO-2013096423-A1 COMBINATION THERAPY WITH INTERFERON AND ANDROGRAPHOLIDES FOR MULTIPLE SCLEROSIS Herbal Powers Corporation (US) 2013-06-27 WO claimed
US-20220409573-A1 Hippocampus Regeneration And Memory Recovery INNOBIOSCIENCE, LLC (US) 2022-12-29 US disclosed
CN-109562097-B Progressive forms of andrographolide for treating multiple sclerosis 因诺生物科学有限责任公司 2022-06-07 CN disclosed
US-10722492-B2 Andrographolide treats progressive forms of multiple sclerosis Inno Bioscience, LLC (US) 2020-07-28 US disclosed
US-20190083458-A1 Andrographolide Treats Progressive Forms of Multiple Sclerosis INNOBIOSCIENCES, LLC (US) 2019-03-21 US disclosed
US-9060994-B2 Combination therapy with interferon and andrographolides for Multiple Sclerosis Inno Biosciences, S.p.A. (CL) 2015-06-23 US disclosed
US-20140301981-A1 Combination Therapy with Interferon and Andrographolides for Multiple Sclerosis INNOBIOSCIENCE LLC (US) 2014-10-09 US disclosed
US-6040449-A USEFUL FOR FORMING FLUORINE CONTAINING 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES, USEFUL AS ANTAGONIST FOR MUSCARINIC M3 RECEPTORS AND LESS SIDE EFFECT BANYU PHARMACEUTICAL CO LTD (JP) 2000-03-21 US disclosed
US-5948792-A POTENT AND SELECTIVE ANTAGONISTS FOR MUSCARINIC M.SUB.3 RECEPTORS WITH LITTLE SIDE EFFECTS. BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US disclosed
EP-0930298-A1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-07-21 EP disclosed