SCHEMBL1994157

SCHEMBL1994157

C=CCc1ccoc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262869 0.78
SCHEMBL6300046 0.77
SCHEMBL16992903 0.77
SCHEMBL8051960 0.76
SCHEMBL8670493 0.73 HCAR2 (0.38)
SCHEMBL357256 0.72
SCHEMBL2840244 0.72
SCHEMBL14877409 0.71
SCHEMBL8670495 0.71 ALOX5 (0.43)
SCHEMBL173301 0.70 ALDH1A1 (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 185 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357578-A1 AIRTIGHT FILM WITH CERAMIC SEALING LAYER AND POLYMER SEALING LAYER Quantum MicroMaterials, Inc. 2023-11-09 US claimed
CN-109790079-A C (the sp of organic zinc reagent and heterocycle (quasi-) halide3)-C(sp2) cross-coupling reaction 香港科技大学 2019-05-21 CN claimed
WO-2018019291-A1 C(SP3)-C(SP2) CROSS-COUPLING REACTION OF ORGANOZINC REAGENTS AND HETEROCYCLIC (PSEUDO)HALIDES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2018-02-01 WO claimed
EP-2196847-B1 ELECTROCHROMIC DISPLAY DEVICE AND METHOD FOR MANUFACTURING THE SAME KURARAY CO (JP) 2013-12-11 EP claimed
US-8519150-B2 π-electron conjugated compound, manufacturing method therefor, and π-electron conjugated polymer obtained using same KURARAY CO., LTD. (JP) 2013-08-27 US claimed
US-8233211-B2 Electrochromic display device and its manufacturing method KURARAY CO., LTD. (JP) 2012-07-31 US claimed
US-20100328751-A1 ELECTROCHROMIC DISPLAY DEVICE AND ITS MANUFACTURING METHOD KURARAY CO., LTD. (JP) 2010-12-30 US claimed
CN-101802700-A Electrochromic display device and method for manufacturing the same KURRARAY CO LTD 2010-08-11 CN claimed
EP-2196847-A1 ELECTROCHROMIC DISPLAY DEVICE AND METHOD FOR MANUFACTURING THE SAME Kuraray Co., Ltd. (JP) 2010-06-16 EP claimed
US-20070167488-A1 Novel therapeutic use LEO PHARMA A/S (DK) 2007-07-19 US claimed
EP-0769947-B1 INDOLINONE COMPOUNDS FOR THE TREATMENT OF DISEASE SUGEN INC (US) 2001-05-02 EP claimed
EP-1066257-A2 HETEROCYLIC CLASSES OF COMPOUNDS FOR THE MODULATING TYROSINE PROTEIN KINASE Sugen, Inc. (US) 2001-01-10 EP claimed
WO-2000038519-A1 3-HETEROARYLIDENYL-2-INDOLINONE COMPOUNDS FOR MODULATING PROTEIN KINASE ACTIVITY AND FOR USE IN CANCER CHEMOTHERAPY SUGEN, INC. (US) 2000-07-06 WO claimed
WO-1999048868-A9 HETEROCYCLIC CLASSES OF COMPOUNDS FOR THE MODULATING TYROSINE PROTEIN KINASE SUGEN INC (US) 2000-04-20 WO claimed
WO-1999048868-A2 HETEROCYCLIC CLASSES OF COMPOUNDS FOR THE MODULATING TYROSINE PROTEIN KINASE SUGEN, INC. (US) 1999-09-30 WO claimed
EP-0769947-A4 INDOLINONE COMPOUNDS FOR THE TREATMENT OF DISEASE SUGEN INC (US) 1998-09-30 EP claimed
US-5792783-A CAPABLE OF MODULATING TYROSINE KINASE SIGNAL TRANSDUCTION IN ORDER TO REGULATE, MODULATE AND/OR INHIBIT ABNORMAL CELL PROLIFERATION SUGEN, INC. (US) 1998-08-11 US claimed
EP-0769947-A1 INDOLINONE COMPOUNDS FOR THE TREATMENT OF DISEASE Sugen, Inc. (US) 1997-05-02 EP claimed
WO-1996040116-A1 INDOLINONE COMPOUNDS FOR THE TREATMENT OF DISEASE SUGEN, INC. (US) 1996-12-19 WO claimed
US-5581192-A Conductive liquid compositions and electrical circuit protection devices comprising conductive liquid compositions EATON CORPORATION (US) 1996-12-03 US claimed