SCHEMBL8054579

SCHEMBL8054579

Cc1nnc(-c2ccccc2O)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.49
GUSB P08236 2/20 0.46
ALOX15 P16050 1/20 0.43
PTGS2 P35354 1/20 0.43
MGAM O43451 1/20 0.41
GAA P10253 1/20 0.41
SI P14410 1/20 0.41
MGAM2 Q2M2H8 1/20 0.41
TRPM8 Q7Z2W7 2/20 0.40
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21091032 0.80 ALDH1A1 (0.51) GAAHPGDMEN1NPC1MAPT
SCHEMBL1207261 0.78 ALDH1A1 (0.52) MGAMGAASIMGAM2HPGD
SCHEMBL18610916 0.78 KDM4E (0.61) GUSBNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL22469017 0.77 GUSB (0.46) HTR2BGUSBALOX15PTGS2MGAM
SCHEMBL11331284 0.77 MGAM (0.67) GUSBMGAMGAASIMGAM2
SCHEMBL14362847 0.77 GUSB (0.56) GUSBHPGDMEN1NPC1RAB9A
SCHEMBL2439298 0.77 ALDH1A1 (0.62) GUSBALOX15HPGDMEN1NPC1
SCHEMBL27639560 0.76 GUSB (0.58) GUSBHPGDMEN1NPC1RAB9A
SCHEMBL27639592 0.76 GUSB (0.55) GUSBHPGDMEN1NPC1RAB9A
SCHEMBL2442712 0.74 HSD11B1 (0.54) HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed