SCHEMBL8055017

SCHEMBL8055017

CN(C)c1nc2cccc(O)c2s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.49
APP P05067 2/20 0.46
ACHE P22303 1/20 0.41
KDM4E B2RXH2 2/20 0.38
RAB9A P51151 3/20 0.37
ALDH1A1 P00352 3/20 0.37
KMT2A Q03164 2/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TSHR P16473 2/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL659152 0.80 HTT (0.40) HTTAPPRAB9AALDH1A1KMT2A
SCHEMBL8052248 0.79 NQO2 (0.47) HTTKDM4ERAB9AALDH1A1KMT2A
SCHEMBL4857995 0.75 APP (0.50) HTTAPPACHEKDM4ERAB9A
SCHEMBL3887904 0.71 RAB9A (0.58) HTTAPPKDM4ERAB9AALDH1A1
SCHEMBL9305472 0.71 APP (0.46) APPACHEKDM4ERAB9AALDH1A1
SCHEMBL74889 0.71 PDPK1 (0.53) HTTAPPACHERAB9AALDH1A1
SCHEMBL9305900 0.71 APP (0.46) APPACHEKDM4ERAB9AALDH1A1
SCHEMBL8054536 0.70 TLR8 (0.46) HTTAPPACHEKDM4ERAB9A
SCHEMBL8051929 0.70 TLR8 (0.46) HTTAPPACHEKDM4ERAB9A
Hydrochloric Acid SCHEMBL28519023 0.69 RAB9A (0.57) HTTAPPKDM4ERAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed