SCHEMBL8052248

SCHEMBL8052248

COc1cccc2nc(N(C)C)sc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.47
RAB9A P51151 5/20 0.46
NPC1 O15118 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
TP53 P04637 2/20 0.46
HPGD P15428 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
MAPT P10636 3/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 7/20 0.42
LMNA P02545 2/20 0.42
CYP3A4 P08684 2/20 0.42
POLB P06746 2/20 0.42
G6PD P11413 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055017 0.79 HTT (0.49) NQO2RAB9ANPC1SMN1; SMN2TP53
SCHEMBL659152 0.77 HTT (0.40) NQO2RAB9ANPC1SMN1; SMN2TP53
SCHEMBL8040045 0.77 NQO2 (0.47) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL2138255 0.76 MEN1 (0.62) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL84829 0.75 CYP3A4 (0.57) NQO2RAB9ANPC1HPGDMAPT
SCHEMBL2748734 0.75 NQO2 (0.46) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL2749006 0.75 ALDH1A1 (0.58) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL6901949 0.74 HSP90AA1 (0.48) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL6691814 0.74 ALDH1A1 (0.47) NQO2RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL8052343 0.72 NPC1 (0.48) NQO2RAB9ANPC1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed