SCHEMBL8056933

SCHEMBL8056933

COC(=O)c1cc(-c2nnn(C[C@H]3CC[C@@H](NC(=O)OC(C)(C)C)CC3)n2)cc(C)n1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 20/20 0.56
MMP3 P08254 2/20 0.50
SLC22A8 Q8TCC7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071049 0.92 MMP13 (0.54) MMP13MMP3SLC22A8
SCHEMBL8066141 0.90 MMP13 (0.53) MMP13MMP3SLC22A8
SCHEMBL8067113 0.89 MMP13 (0.56) MMP13MMP3SLC22A8
SCHEMBL3758118 0.87 MMP13 (0.42) MMP13MMP3
SCHEMBL3758113 0.87 MMP13 (0.42) MMP13MMP3
SCHEMBL3798392 0.84 MMP13 (0.68) MMP13MMP3SLC22A8
SCHEMBL3808963 0.84 MMP13 (0.66) MMP13MMP3SLC22A8
SCHEMBL8068202 0.84 MMP13 (0.66) MMP13MMP3SLC22A8
SCHEMBL3808968 0.84 MMP13 (0.66) MMP13MMP3SLC22A8
SCHEMBL3798394 0.84 MMP13 (0.68) MMP13MMP3SLC22A8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed