SCHEMBL8057294

SCHEMBL8057294

COC(=O)c1cc2c(cc1C(F)(F)F)C=C(C)S2(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CFTR P13569 7/20 0.41
NOTUM Q6P988 4/20 0.40
MAPT P10636 3/20 0.36
SOS1 Q07889 1/20 0.34
MBOAT4 Q96T53 1/20 0.34
ALDH1A1 P00352 2/20 0.31
HSD17B10 Q99714 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
ATM Q13315 1/20 0.31
KDR P35968 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
P4HB P07237 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060827 0.82 KDM4E (0.33) CFTRNOTUMMAPTSOS1ALDH1A1
SCHEMBL8045255 0.81 KDM4E (0.38) MAPTALDH1A1HSD17B10KDM4EGLA
SCHEMBL8057300 0.78 CFTR (0.46) CFTRNOTUMMAPTSOS1ALDH1A1
SCHEMBL8057109 0.78 ALDH1A1 (0.34) MAPTALDH1A1HSD17B10KDM4EGLA
SCHEMBL8057039 0.76 CFTR (0.41) CFTRNOTUMMAPTSOS1MBOAT4
SCHEMBL8062894 0.72 CFTR (0.40) CFTRNOTUMMAPTSOS1P4HB
SCHEMBL8056417 0.71 CFTR (0.39) CFTRNOTUMMAPTSOS1
SCHEMBL8056939 0.71 CA1 (0.46) NOTUMMAPTALDH1A1HSD17B10KDM4E
SCHEMBL8062790 0.70 NOTUM (0.43) CFTRNOTUMMAPTSOS1
SCHEMBL24983697 0.70 CFTR (0.51) CFTRNOTUMMAPTSOS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed