SCHEMBL8058080

SCHEMBL8058080

COC(=O)c1cc2c(cc1F)C(C)=CS2(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
ALPL P05186 2/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KDM4E B2RXH2 5/20 0.33
HSD17B10 Q99714 4/20 0.33
MAPT P10636 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
ILK Q13418 1/20 0.33
CYP46A1 Q9Y6A2 1/20 0.32
CA12 O43570 2/20 0.32
CA7 P43166 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057039 0.82 CFTR (0.41) CA1CA2CA9KDM4EHSD17B10
SCHEMBL8058137 0.81 ALDH1A1 (0.36) CA1CA2CA9KDM4EHSD17B10
SCHEMBL8056463 0.74 CA1 (0.50) CA1CA2CA9KDM4EHSD17B10
SCHEMBL522786 0.73 CA12 (0.47) CA1CA2CA9SLC6A4SLC6A3
SCHEMBL8058193 0.72 VEGFA (0.41) CA1CA2CA9ALPLSLC6A4
SCHEMBL8058094 0.71 ALDH1A1 (0.33) CA1CA2CA9ALPLSLC6A4
SCHEMBL8060827 0.71 KDM4E (0.33) CA1CA2CA9SLC6A4SLC6A3
SCHEMBL19993672 0.70 MAPT (0.42) CA1CA2CA9SLC6A4SLC6A3
SCHEMBL8056507 0.70 CTSL (0.36) ALPLSLC6A4SLC6A3KDM4EHSD17B10
SCHEMBL8056511 0.70 CTSL (0.36) ALPLSLC6A4SLC6A3KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed