SCHEMBL8058149

SCHEMBL8058149

C=C1CS(=O)(=O)c2cc(C(=O)OC)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA12 O43570 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
XDH P47989 1/20 0.44
PTPRC P08575 1/20 0.42
PDK2 Q15119 2/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
ATM Q13315 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8258364 0.83 CA1 (0.45) CA1CA2CA12CA7CA9
SCHEMBL5904274 0.83 PTPRC (0.47) CA1CA2CA12CA7CA9
SCHEMBL13593187 0.79 CA12 (0.41) CA1CA2CA12CA7CA9
SCHEMBL8060698 0.79 KDM4E (0.36) CA1CA2CA12CA7CA9
SCHEMBL10164105 0.79 CA12 (0.41) CA1CA2CA12CA7CA9
SCHEMBL8058159 0.78 CA12 (0.41) CA1CA2CA12CA7CA9
SCHEMBL8058154 0.78 CA12 (0.41) CA1CA2CA12CA7CA9
SCHEMBL8058094 0.75 ALDH1A1 (0.33) CA1CA2CA12CA7CA9
SCHEMBL8058155 0.75 HTR2B (0.47)
SCHEMBL15398420 0.75 CA1 (0.53) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed