SCHEMBL8058181

SCHEMBL8058181

COC(=O)c1ccc2c(c1)S(=O)(=O)C(C)(C)O2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.46
CA12 O43570 4/20 0.44
CA9 Q16790 4/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA7 P43166 2/20 0.44
CA14 Q9ULX7 2/20 0.44
XDH P47989 1/20 0.44
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
LCK P06239 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060643 0.79 KDM4E (0.36) ALOX5CA12CA9CA1CA2
SCHEMBL8045354 0.78 ALOX5 (0.43) ALOX5CA12CA9CA1CA2
SCHEMBL8056352 0.78 RARB (0.46) ALOX5CA12CA9CA1CA2
SCHEMBL13822771 0.78 KMT2A (0.36) ALDH1A1HSD17B10GAASMN1; SMN2MEN1
SCHEMBL8058203 0.75 CA12 (0.41) ALOX5CA12CA9CA1CA2
SCHEMBL24401018 0.74 ALOX5 (0.50) ALOX5CA12CA9CA1CA2
SCHEMBL13822626 0.72 LMNA (0.44) GAALMNARAB9A
SCHEMBL13822628 0.72 LMNA (0.44) GAALMNARAB9A
SCHEMBL8062909 0.72 CA1 (0.42) ALOX5CA12CA9CA1CA2
SCHEMBL8056514 0.71 NPC1 (0.45) ALOX5CA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed