SCHEMBL8058546

SCHEMBL8058546

C/C(=C\c1cc(F)cc(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.44
RXRA P19793 2/20 0.41
RXRB P28702 2/20 0.41
RXRG P48443 2/20 0.41
RPS6KA3 P51812 1/20 0.41
JAK3 P52333 1/20 0.41
ACKR3 P25106 2/20 0.37
GPR35 Q9HC97 2/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
PTGS1 P23219 1/20 0.36
CES2 O00748 1/20 0.35
NR4A1 P22736 1/20 0.35
NR4A2 P43354 1/20 0.35
NR4A3 Q92570 1/20 0.35
APEX1 P27695 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
TBXAS1 P24557 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058552 1.00 AKR1C3 (0.44) AKR1C3RXRARXRBRXRGRPS6KA3
SCHEMBL7133171 0.84 AKR1C3 (0.55) AKR1C3PTGS1CES2APEX1TBXAS1
SCHEMBL7133176 0.84 AKR1C3 (0.55) AKR1C3PTGS1CES2APEX1TBXAS1
Guanidine SCHEMBL8058713 0.81 RPS6KA3 (0.49) AKR1C3RXRARXRBRXRGRPS6KA3
SCHEMBL8042956 0.77 AKR1C3 (0.58) AKR1C3LMNAMAPTHPGDCES2
SCHEMBL5004361 0.77 AKR1C3 (0.58) AKR1C3LMNAMAPTHPGDCES2
SCHEMBL12498144 0.76 AKR1C3 (0.43) AKR1C3RXRARXRBRXRGLMNA
SCHEMBL12498149 0.76 AKR1C3 (0.43) AKR1C3RXRARXRBRXRGLMNA
SCHEMBL6933101 0.76 AKR1C3 (0.60) AKR1C3PTGS1CES2NR4A1NR4A2
SCHEMBL6933104 0.76 AKR1C3 (0.60) AKR1C3PTGS1CES2NR4A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6025349-A ANTIARRHYTHMIC PROPERTIES, HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-15 US disclosed