SCHEMBL8060271

SCHEMBL8060271

CCCCc1nc(Cc2ccc(-c3ccccc3C(=O)O)cc2)c(C=O)[nH]1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 7/20 0.59
AGTR1 P30556 1/20 0.55
AGTR2 P50052 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6534730 0.81 BRS3 (0.52) BRS3AGTR1AGTR2
SCHEMBL9196627 0.78 AGTR1 (0.55) BRS3AGTR1AGTR2
SCHEMBL9304542 0.78 BRS3 (0.56) BRS3AGTR1AGTR2
SCHEMBL9200834 0.78 AGTR1 (0.53) BRS3AGTR1AGTR2
SCHEMBL1227544 0.77 BRS3 (0.55) BRS3AGTR1AGTR2
SCHEMBL9428665 0.76 AGTR1 (0.55) BRS3AGTR1AGTR2
SCHEMBL9552678 0.76 BRS3 (0.57) BRS3AGTR1AGTR2
SCHEMBL9510826 0.76 BRS3 (0.55) BRS3AGTR1AGTR2
SCHEMBL9452733 0.76 BRS3 (0.56) BRS3AGTR1AGTR2
SCHEMBL3906504 0.76 BRS3 (0.70) BRS3AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962500-A HYPOSENSITVE AGENT MERCK SHARP & DOHME CORP. 1999-10-05 US claimed
EP-0533840-A1 TREATMENT OF CHRONIC RENAL FAILURE WITH IMIDAZOLE ANGIOTENSIN-II RECEPTOR ANTAGONISTS. DU PONT (US) 1993-03-31 EP claimed
EP-1019048-A1 USE OF AN ANGIOTENSIN II RECEPTOR ANTAGONIST FOR THE PREPARATION OF DRUGS TO INCREASE THE SURVIVAL RATE OF RENAL TRANSPLANT PATIENTS Merck Sharp Dohme (Italia) S.P.A. (IT) 2000-07-19 EP disclosed
US-5962500-A HYPOSENSITVE AGENT MERCK SHARP & DOHME CORP. 1999-10-05 US disclosed
WO-1999016437-A1 USE OF AN ANGIOTENSIN II RECEPTOR ANTAGONIST FOR THE PREPARATION OF DRUGS TO INCREASE THE SURVIVAL RATE OF RENAL TRANSPLANT PATIENTS MERCK SHARP DOHME (ITALIA) S.P.A. (IT) 1999-04-08 WO disclosed
US-5663186-A TREATING ATHEROSCLEROSIS AND REDUCING CHOLESTEROL ALONE OR IN CONJUCTION WITH THE TREATMENT OF HYPERTENSION USING A MIXTURE OF LOSARTAN, SIMVASTATIN AND ENALPRIL MERCK & CO., INC. (US) 1997-09-02 US disclosed