SCHEMBL8060736

SCHEMBL8060736

CS(=O)(=O)Cl.O=C(NCc1ccc(Cl)c(Cl)c1)c1cc2ccccc2[nH]1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 2/20 0.54
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54
NCOR2 Q9Y618 1/20 0.54
DRD2 P14416 1/20 0.51
DRD3 P35462 1/20 0.51
NAMPT P43490 2/20 0.50
CYP2C9 P11712 1/20 0.50
HTR2C P28335 1/20 0.50
NHERF1 O14745 1/20 0.50
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 2/20 0.49
GAA P10253 1/20 0.49
MAPK1 P28482 1/20 0.49
SRC P12931 1/20 0.48
HSD17B10 Q99714 1/20 0.48
IDO1 P14902 1/20 0.48
CNR1 P21554 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300914 0.93 HDAC2 (0.57) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL18750641 0.85 HDAC2 (0.57) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL17149766 0.83 HDAC2 (0.57) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL6657894 0.81 NHERF1 (0.69) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL17149769 0.79 LMNA (0.62) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL2760063 0.78 HDAC3 (0.60) HDAC2HDAC3HDAC1NAMPTCYP2C9
SCHEMBL2735969 0.78 CA12 (0.72) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL6885836 0.77 HDAC2 (0.59) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL18669175 0.77 KDM4E (0.60) HDAC2HDAC3HDAC1DRD2DRD3
SCHEMBL6657027 0.77 HDAC2 (0.67) HDAC2HDAC3HDAC1NCOR2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-A2 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS AstraZeneca UK Limited (GB) 2000-05-31 EP disclosed
WO-1999007351-A2 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ZENECA LIMITED (GB) 1999-02-18 WO disclosed