SCHEMBL8060757

SCHEMBL8060757

COC(=O)c1cc2c(cc1C)N(C)CS2(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.37
ALDH1A1 P00352 6/20 0.37
CASP1 P29466 2/20 0.37
CASP7 P55210 2/20 0.37
HSD17B10 Q99714 2/20 0.37
ALOX15 P16050 1/20 0.37
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
GLA P06280 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 3/20 0.35
MYC P01106 1/20 0.34
CASP3 P42574 1/20 0.34
POLB P06746 1/20 0.34
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057305 0.86 ALDH1A1 (0.41) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8062935 0.79 ALDH1A1 (0.51) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8045290 0.79 ALDH1A1 (0.38) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8062771 0.79 ALDH1A1 (0.36) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8060788 0.79 ALDH1A1 (0.36) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8057283 0.73 PDGFRB (0.36) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8056874 0.73 ALDH1A1 (0.35) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8056444 0.71 ALDH1A1 (0.36) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8063021 0.71 LMNA (0.40) KDM4EALDH1A1CASP1CASP7HSD17B10
SCHEMBL8056369 0.70 ALDH1A1 (0.39) KDM4EALDH1A1CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed