SCHEMBL8060993

SCHEMBL8060993

FC(F)(F)c1cc(Cl)c2cc(COc3cc[c]cc3)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.49
EGFR P00533 1/20 0.47
EPHA2 P29317 1/20 0.47
KDR P35968 1/20 0.47
EPHB4 P54760 1/20 0.47
PPARG P37231 16/20 0.41
TEC P42680 1/20 0.38
PTGES O14684 1/20 0.37
ALOX5 P09917 1/20 0.37
PSEN1 P49768 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12301252 0.81 EGFR (0.48) NT5EEGFREPHA2KDREPHB4
SCHEMBL4050447 0.76 ADAM17 (0.49)
SCHEMBL14591907 0.74 NT5E (0.60) NT5EEGFREPHA2KDREPHB4
SCHEMBL485686 0.74 NT5E (0.65) NT5EEGFREPHA2KDREPHB4
SCHEMBL11955074 0.72 NT5E (0.57) NT5EEGFREPHA2KDREPHB4
SCHEMBL27766191 0.72 NT5E (0.61) NT5EEGFREPHA2KDREPHB4
SCHEMBL14307070 0.72 NT5E (0.57) NT5EEGFREPHA2KDREPHB4
SCHEMBL4900145 0.71 THRA (0.60) NT5EEGFREPHA2KDREPHB4
SCHEMBL693400 0.71 NT5E (0.55) NT5E
SCHEMBL13197081 0.71 NT5E (0.56) NT5EEGFREPHA2KDREPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057336-A ANTIINFLAMMATORY AGENTS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-05-02 US disclosed