SCHEMBL8062875

SCHEMBL8062875

CC1Cc2ccc(C(=O)N=C(N)N)cc2S(=O)(=O)C1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.45
HTR2B P41595 3/20 0.45
DRD2 P14416 1/20 0.45
ADRA1D P25100 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
SLC9A1 P19634 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062978 0.87 HTR2B (0.45) HTR7HTR2BDRD2ADRA1DHTR2A
SCHEMBL8060822 0.83 HTR2B (0.46) HTR7HTR2BDRD2ADRA1DHTR2A
SCHEMBL8056274 0.83 HTR2B (0.46) HTR7HTR2B
SCHEMBL8045289 0.81
SCHEMBL8045075 0.78 HTR2B (0.48) HTR7HTR2B
SCHEMBL8045374 0.78 HTR2B (0.46) HTR7HTR2B
SCHEMBL8058186 0.78 HTR7 (0.49) HTR7HTR2BDRD2ADRA1DHTR2A
SCHEMBL8045091 0.78 ALDH1A1 (0.45)
SCHEMBL8045040 0.77 HTR2B (0.44) HTR7HTR2B
SCHEMBL8045272 0.77 HTR7 (0.41) HTR7HTR2BSLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed