SCHEMBL8063451

SCHEMBL8063451

CC(CC(C)(C)C)C(NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)CNC(=O)c1csc(NC(=O)NCc2ccccc2)n1)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.37
ROCK1 Q13464 5/20 0.37
PSMB8 P28062 2/20 0.36
PSMB5 P28074 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
BACE1 P56817 4/20 0.34
LCK P06239 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGAV P06756 2/20 0.34
PSMB11 A5LHX3 1/20 0.34
PSMA7 O14818 1/20 0.34
PSMB1 P20618 1/20 0.34
PSMA1 P25786 1/20 0.34
PSMA2 P25787 1/20 0.34
PSMA3 P25788 1/20 0.34
PSMA4 P25789 1/20 0.34
PSMB9 P28065 1/20 0.34
PSMA5 P28066 1/20 0.34
PSMB4 P28070 1/20 0.34
PSMB6 P28072 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7139835 0.93 ROCK2 (0.39) ROCK2ROCK1PSMB8PSMB5BACE1
SCHEMBL7139827 0.93 ROCK2 (0.39) ROCK2ROCK1PSMB8PSMB5BACE1
SCHEMBL8063448 0.89 ROCK2 (0.39) ROCK2ROCK1PSMB8PSMB5BACE1
SCHEMBL27510568 0.89 ROCK2 (0.39) ROCK2ROCK1PSMB8PSMB5BACE1
SCHEMBL8063417 0.89 ROCK2 (0.43) ROCK2ROCK1PSMB8PSMB5SMN1; SMN2
SCHEMBL8062348 0.88 ROCK2 (0.41) ROCK2ROCK1PSMB8PSMB5SMN1; SMN2
SCHEMBL8051508 0.86 ROCK2 (0.43) ROCK2ROCK1SMN1; SMN2ITGB3ITGAV
SCHEMBL8051485 0.85 ROCK2 (0.39) ROCK2ROCK1PSMB8PSMB5SMN1; SMN2
SCHEMBL8063461 0.84 ROCK2 (0.38) ROCK2ROCK1PSMB8PSMB5SMN1; SMN2
SCHEMBL8063457 0.84 ROCK2 (0.38) ROCK2ROCK1PSMB8PSMB5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100282-A Thiazole derivatives HOFFMAN-LA ROCHE INC. (US) 2000-08-08 US disclosed