SCHEMBL806481

SCHEMBL806481

CCc1c(C)c(C)cc2cc(C#N)n(C)c12

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
MDM2 Q00987 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KDM5A P29375 1/20 0.31
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
MEN1 O00255 1/20 0.30
HK1 P19367 1/20 0.30
KMT2A Q03164 1/20 0.30
HKDC1 Q2TB90 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24629878 0.69 AR (0.41) ARSMN1; SMN2KDM4EMEN1KMT2A
SCHEMBL26581297 0.68 TSHR (0.38) ARNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL13767120 0.66 KDM4E (0.42) NPC1LMNAMAPTRAB9AMDM2
SCHEMBL12320911 0.63 AR (0.36) ARMEN1KMT2A
SCHEMBL9461239 0.63 PGK1 (0.36) TSHR
SCHEMBL13735112 0.63 KMT2A (0.42) ARKDM4EUSP2MEN1KMT2A
SCHEMBL24629973 0.62 MEN1 (0.33) ARMEN1KMT2A
SCHEMBL24392772 0.62 KDM4E (0.40) ARLMNAMAPTNPSR1KDM4E
SCHEMBL806475 0.62 RXFP1 (0.49) ARNPC1LMNAMAPTRAB9A
SCHEMBL29769066 0.62 RXFP1 (0.49) ARNPC1LMNAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036253-A1 HETEROCYCLIC COMPOUNDS FOR TREATING OR PREVENTING DISORDERS CAUSED BY REDUCED NEUROTRANSMISSION OF SEROTONIN, NOREPHNEPHRINE OR DOPAMINE. OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-03-22 WO disclosed