SCHEMBL806482

SCHEMBL806482

Cc1cc2ccc(O)cc2c(C)c1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.43
ESR2 Q92731 8/20 0.43
HSD17B3 P37058 2/20 0.43
MCL1 Q07820 1/20 0.40
PTGES O14684 1/20 0.40
CYP1A2 P05177 1/20 0.38
ACHE P22303 1/20 0.38
TLR8 Q9NR97 1/20 0.38
DYRK1A Q13627 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13316750 0.85 ESR1 (0.42) ESR1ESR2HSD17B3MCL1PTGES
SCHEMBL12856652 0.79 ESR1 (0.41) ESR1ESR2HSD17B3MCL1PTGES
SCHEMBL23322803 0.77 CYP1A2 (0.50) CYP1A2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2209442 0.76 ESR1 (0.58) ESR1ESR2MCL1CYP1A2TLR8
SCHEMBL29771841 0.76 ESR1 (0.58) ESR1ESR2MCL1CYP1A2TLR8
SCHEMBL9623383 0.76 ESR2 (0.52) ESR1ESR2MCL1CYP1A2TLR8
SCHEMBL12912891 0.75 ESR1 (0.46) ESR1ESR2HSD17B3MCL1PTGES
SCHEMBL29276380 0.75 CYP1A2 (0.45) ESR2HSD17B3MCL1CYP1A2KDM4E
SCHEMBL2046089 0.74 ESR1 (0.52) ESR1ESR2HSD17B3MCL1CYP1A2
SCHEMBL806516 0.74 CYP1A2 (0.54) ESR1ESR2MCL1PTGESCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8303844-B2 Benzo[f]chrome any pyrano[3,2-f]chrome derivatives for use in liquid crystal media MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2012-11-06 US disclosed
WO-2012036253-A1 HETEROCYCLIC COMPOUNDS FOR TREATING OR PREVENTING DISORDERS CAUSED BY REDUCED NEUROTRANSMISSION OF SEROTONIN, NOREPHNEPHRINE OR DOPAMINE. OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2012-03-22 WO disclosed
US-20110043746-A1 BENZO[F]CHROME ANY PYRANO[3,2-F]CHROME DERIVATIVES FOR USE IN LIQUID CRYSTAL MEDIA MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110043746-A1 BENZO[F]CHROME ANY PYRANO[3,2-F]CHROME DERIVATIVES FOR USE IN LIQUID CRYSTAL MEDIA CHRM1, F12, CTRB2 ESR1 360/4885ESR2 589/4885HSD17B3 2110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.