SCHEMBL8065402

SCHEMBL8065402

COc1cccc(CNC(=O)c2cc(-c3ncn(CC4CCC(N)CC4)n3)nc(C)n2)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 17/20 0.55
MMP3 P08254 2/20 0.52
KDM4E B2RXH2 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3806955 0.91 MMP13 (0.56) MMP13MMP3KDM4EHSD17B10ROCK2
SCHEMBL8066650 0.89 MMP13 (0.55) MMP13MMP3KDM4EHSD17B10ROCK2
SCHEMBL8063937 0.88 MMP13 (0.66) MMP13MMP3
SCHEMBL8065798 0.87 MMP13 (0.53) MMP13MMP3KDM4EHSD17B10ROCK2
SCHEMBL8070773 0.86 MMP13 (0.54) MMP13MMP3KDM4EHSD17B10ROCK2
SCHEMBL8074480 0.86 MMP13 (0.56) MMP13ROCK2ROCK1
SCHEMBL3804778 0.86 MMP13 (0.71) MMP13MMP3
SCHEMBL3805005 0.86 MMP13 (0.71) MMP13MMP3
SCHEMBL3747906 0.83 MMP13 (0.76) MMP13MMP3KDM4EHSD17B10ROCK1
SCHEMBL3747903 0.83 MMP13 (0.76) MMP13MMP3KDM4EHSD17B10ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed