SCHEMBL8065405

SCHEMBL8065405

O=C(NCCc1cccc2ccccc12)C1CC1

nearest known ligand 0.89

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 0.67
MTNR1B P49286 6/20 0.66
NQO2 P16083 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6254856 0.94 MTNR1A (0.69) MTNR1AMTNR1BNQO2
SCHEMBL9131349 0.93 MTNR1A (0.69) MTNR1AMTNR1BNQO2
SCHEMBL14615455 0.91 MTNR1A (0.61) MTNR1AMTNR1BNQO2
SCHEMBL5339923 0.85 MTNR1A (0.71) MTNR1AMTNR1BNQO2
SCHEMBL27450734 0.82 MTNR1A (0.70) MTNR1AMTNR1BNQO2
SCHEMBL8065738 0.81 MTNR1A (0.52) MTNR1AMTNR1BNQO2
SCHEMBL8961285 0.81 MTNR1A (0.56) MTNR1AMTNR1BNQO2
SCHEMBL6075677 0.81 MTNR1A (0.72) MTNR1AMTNR1BNQO2
SCHEMBL6247137 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL29493844 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562956-B1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-09-27 EP claimed
US-5420158-A Melatonin activity ADIR ET COMPAGNIE (FR) 1995-05-30 US claimed
EP-0562956-A1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-09-29 EP claimed
JP-6049011-A None JP disclosed
CN-1155562-C Novel naphthalene compounds, process for their preparation and pharmaceutical compositions containing them ɪά��ʵ���� 2004-06-30 CN disclosed
US-6143789-A ENANTIOMORPHS ADIR ET COMPAGNIE (FR) 2000-11-07 US disclosed
CN-1221734-A Novel naphthalene compounds, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1999-07-07 CN disclosed
EP-0919541-A1 Naphthalene compounds, process for their preparation and their pharmaceutical compositions ADIR ET COMPAGNIE (FR) 1999-06-02 EP disclosed
US-5616614-A USEFUL IN TREATMENT OF DISORDERS LINKED TO ABNORMAL MELATONIN ACTIVITY ADIR ET COMPAGNIE (FR) 1997-04-01 US disclosed
EP-0562956-B1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-09-27 EP disclosed
US-5420158-A Melatonin activity ADIR ET COMPAGNIE (FR) 1995-05-30 US disclosed
JP-H0649011-A NEW NAPHTHYLALKYLAMINE, ITS PREPARATION AND PHERMACEUTICAL COMPOSITION CONTAINING THE SAME ADIR 1994-02-22 JP disclosed
EP-0562956-A1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-09-29 EP disclosed