SCHEMBL8065853

SCHEMBL8065853

NCc1cncc(CN)n1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 8/20 0.36
AOC1 P19801 3/20 0.36
LOXL2 Q9Y4K0 2/20 0.33
HRH4 Q9H3N8 1/20 0.31
CDK2 P24941 1/20 0.31
CYP2A6 P11509 2/20 0.30
MAOA P21397 1/20 0.30
LOX P28300 1/20 0.30
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5751670 0.82
SCHEMBL346239 0.82
Hydrochloric Acid SCHEMBL2673701 0.80 AOC3 (0.38) AOC3AOC1
SCHEMBL946103 0.77 LOXL2 (0.36) AOC3AOC1LOXL2LOX
SCHEMBL214832 0.69
SCHEMBL11870165 0.69 CCR1 (0.42)
SCHEMBL522024 0.69 HRH4 (0.46) LOXL2HRH4MAOAGRIN2DGRIN3B
SCHEMBL830961 0.69 NOS3 (0.36) AOC3HRH4GRIN2DGRIN3BGRIN1
Hydrochloric Acid SCHEMBL707452 0.67 HSP90AA1 (0.44) AOC3AOC1LOXL2CYP2A6
Hydrochloric Acid SCHEMBL5121 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001944-A1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2000-05-24 EP claimed
WO-1999003844-A1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1999-01-28 WO claimed
EP-1001944-A1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2000-05-24 EP disclosed
WO-1999003844-A1 PYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1999-01-28 WO disclosed