SCHEMBL8067896

SCHEMBL8067896

CC(C)(OC(=O)C12CC3CC(CC(C3)C1)C2)c1cccnc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 1.00
CYP17A1 P05093 12/20 1.00
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HSD11B1 P28845 2/20 0.47
P2RX7 Q99572 1/20 0.47
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8067904 0.84 CYP17A1 (1.00) CYP19A1CYP17A1MEN1KMT2AALDH1A1
SCHEMBL9334979 0.74 CYP19A1 (1.00) CYP19A1CYP17A1HSD11B1
SCHEMBL31239310 0.72 CYP19A1 (0.56) CYP19A1CYP17A1MEN1KMT2AALDH1A1
SCHEMBL8899923 0.72 CYP17A1 (1.00) CYP19A1CYP17A1MEN1KMT2AHSD11B1
SCHEMBL8897307 0.72 CYP17A1 (1.00) CYP19A1CYP17A1MEN1KMT2AHSD11B1
SCHEMBL8897312 0.72 CYP17A1 (1.00) CYP19A1CYP17A1MEN1KMT2AHSD11B1
SCHEMBL8077869 0.71 CYP17A1 (1.00) CYP19A1CYP17A1MEN1KMT2AHSD11B1
SCHEMBL23746946 0.70 CYP19A1 (0.53) CYP19A1CYP17A1KMT2AALDH1A1
SCHEMBL25899389 0.69 CYP19A1 (0.52) CYP19A1CYP17A1ALDH1A1
SCHEMBL131064 0.69 CYP17A1 (0.55) CYP19A1CYP17A1MEN1KMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640072-B1 Derivatives of pyridine as hydroxylase and lyase inhibitors BTG INT LTD (GB) 2000-08-23 EP disclosed
US-5595995-A ANTICARCINOGENIC AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-01-21 US disclosed
EP-0640072-A1 SUBSTITUTED PYRIDINES, THEIR PREPARATION AND PHARMACEUTICAL USE BTG INTERNATIONAL LIMITED (GB) 1995-03-01 EP disclosed
WO-1993023375-A1 SUBSTITUTED PYRIDINES, THEIR PREPARATION AND PHARMACEUTICAL USE BRITISH TECHNOLOGY GROUP LIMITED (GB) 1993-11-25 WO disclosed