SCHEMBL8077869

SCHEMBL8077869

O=C(OCc1cccnc1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 9/20 1.00
CYP19A1 P11511 9/20 1.00
HSD11B1 P28845 2/20 0.69
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
P2RX7 Q99572 2/20 0.53
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
LMNA P02545 1/20 0.50
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8075850 0.83 CYP19A1 (1.00) CYP17A1CYP19A1HSD11B1MEN1KMT2A
SCHEMBL1733254 0.83 CYP17A1 (0.73) CYP17A1CYP19A1HSD11B1P2RX7ALDH1A1
SCHEMBL3321259 0.82 HSD11B1 (1.00) CYP17A1CYP19A1HSD11B1MEN1KMT2A
Trimethylammonium SCHEMBL7978797 0.78 CYP17A1 (0.66) CYP17A1CYP19A1HSD11B1MEN1KMT2A
SCHEMBL1770008 0.77 HSD11B1 (0.67) CYP17A1CYP19A1HSD11B1MEN1KMT2A
SCHEMBL31613300 0.76 CYP17A1 (0.63) CYP17A1CYP19A1KMT2AALDH1A1CYP1A2
SCHEMBL21082070 0.76 CYP17A1 (0.61) CYP17A1CYP19A1HSD11B1MEN1KMT2A
SCHEMBL13333015 0.76 CYP17A1 (1.00) CYP17A1CYP19A1HSD11B1MEN1KMT2A
SCHEMBL31538453 0.75 CYP17A1 (0.66) CYP17A1CYP19A1MEN1KMT2AP2RX7
SCHEMBL20620855 0.75 CYP17A1 (0.60) CYP17A1CYP19A1HSD11B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640072-B1 Derivatives of pyridine as hydroxylase and lyase inhibitors BTG INT LTD (GB) 2000-08-23 EP disclosed
US-5595995-A ANTICARCINOGENIC AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-01-21 US disclosed