SCHEMBL8068441

SCHEMBL8068441

CC(c1c[nH]c2ccccc12)[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NMBR P28336 3/20 0.58
MAPT P10636 4/20 0.53
HTT P42858 2/20 0.53
GAA P10253 1/20 0.53
CASP1 P29466 1/20 0.52
LMNA P02545 3/20 0.52
TACR1 P25103 1/20 0.50
SSTR1 P30872 1/20 0.49
BMP1 P13497 1/20 0.48
MME P08473 2/20 0.48
ECE1 P42892 2/20 0.48
MMP9 P14780 2/20 0.48
MMP8 P22894 2/20 0.48
MMP2 P08253 1/20 0.48
MMP14 P50281 1/20 0.48
ALDH1A1 P00352 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8700867 1.00 NMBR (0.58) NMBRMAPTHTTGAACASP1
SCHEMBL8706625 0.84 NMBR (0.49) NMBRMAPTHTTGAACASP1
SCHEMBL5913306 0.82 CTSL (0.53) MAPTTACR1SSTR1SMN1; SMN2
SCHEMBL8528011 0.82 CTSL (0.53) MAPTTACR1SSTR1SMN1; SMN2
SCHEMBL27621167 0.82 CTSL (0.53) MAPTTACR1SSTR1SMN1; SMN2
SCHEMBL8022191 0.82 CTSL (0.53) MAPTTACR1SSTR1SMN1; SMN2
SCHEMBL31000751 0.81 MDM4 (0.46)
SCHEMBL31000753 0.81 MDM4 (0.46)
SCHEMBL6480706 0.81 MDM4 (0.46)
SCHEMBL6481998 0.81 MDM4 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030983-A ANTITUMOR AND -CARCINOGENIC AGENTS; ANTIBIOTICS; BACTERICIDES; VIRICIDES; PARACITICIDES; ENZYME INHIBITORS; POLYMERASES; FARNESYL-PROTEIN TRANSFERASE; RAS PROTEINS BALL STATE UNIVERSITY (US) 2000-02-29 US disclosed
US-6025372-A Somatostatin agonists MERCK & CO., INC. (US) 2000-02-15 US disclosed
US-5712289-A ANTITUMOR AGENTS, INTERMEDIATES FOR LAVENDAMYCINS BALL STATE UNIVERSITY (US) 1998-01-27 US disclosed
US-5646150-A ADMINISTERING AS ANTITUMOR AGENT, ANTIPROTOZOA AGENT, VIRICIDE, PARASITICIDE, OR BACTERICIDE BALL STATE UNIVERSITY (US) 1997-07-08 US disclosed
US-5525611-A ANTITUMOR AGENT, BACTERICIDES, VIRICIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 1996-06-11 US disclosed
WO-1994029308-A1 LAVENDAMYCIN ANALOGS, THEIR USE AND PREPARATION BEHFOROUZ MOHAMMAD (US) 1994-12-22 WO disclosed