SCHEMBL8069682

SCHEMBL8069682

CN(C)CCN(C)CC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA2 P00918 1/20 0.56
CA3 P07451 1/20 0.56
CA4 P22748 1/20 0.56
CA6 P23280 1/20 0.56
CA5A P35218 1/20 0.56
CA7 P43166 1/20 0.56
CA9 Q16790 1/20 0.56
CA14 Q9ULX7 1/20 0.56
CA5B Q9Y2D0 1/20 0.56
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
TNNI3 P19429 1/20 0.33
TNNT2 P45379 1/20 0.33
TNNC1 P63316 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29581038 0.88 CA12 (0.44) CA12CA2CA3CA4CA6
SCHEMBL29581876 0.88 CA12 (0.44) CA12CA2CA3CA4CA6
SCHEMBL27100952 0.83 ALDH1A1 (0.50) CA12CA2CA3CA4CA6
SCHEMBL28091491 0.80 TDP1 (0.45) CA12CA2CA3CA4CA6
SCHEMBL25853689 0.79 CA12 (0.33) CA12CA2CA3CA4CA6
SCHEMBL30664066 0.78 CA12 (0.50) CA12CA2CA3CA4CA6
SCHEMBL16821921 0.78 CA12 (0.50) CA12CA2CA3CA4CA6
SCHEMBL4120760 0.77 TSHR (0.33) TSHRTDP1
SCHEMBL13407589 0.77
SCHEMBL9284840 0.77 TSHR (0.32) TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210283138-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2021-09-16 US disclosed
WO-2020024932-A1 METHOD FOR TREATING CANCER BY COMBINATION OF IAP INHIBITOR AND MODULATOR OF IMMUNE CHECKPOINT MOLECULE ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2020-02-06 WO disclosed
US-20170283398-A1 2-AMINOPYRIMIDINE COMPOUND AND PHARMACEUTICAL COMPOSITION AND USE THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-10-05 US disclosed
US-20140221334-A1 KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-08-07 US disclosed
WO-2014081946-A2 METHODS FOR THE RECYCLING OF WIRE-SAW CUTTING FLUID MEMC SINGAPORE PTE, LTD. (SG) 2014-05-30 WO disclosed
WO-2014081960-A2 SYSTEMS FOR THE RECYCLING OF WIRE-SAW CUTTING FLUID MEMC SINGAPORE PTE, LTD. (SG) 2014-05-30 WO disclosed
US-7879808-B2 potent activity against resistant pneumococci; for treating domestic fowl MEIJI SEIKA KAISHA, LTD. (JP) 2011-02-01 US disclosed
US-20100210570-A1 LINCOMYCIN DERIVATIVES AND ANTIMICROBIAL AGENTS COMPRISING THE SAME AS ACTIVE INGREDIENT MEIJI SEIKA KAISHA LTD. (JP) 2010-08-19 US disclosed
US-20100197908-A1 Pyridazine Derivatives with MCH Antagonistic Activity and Medicaments Comprising These Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-05 US disclosed
US-20100197908-A1 Pyridazine Derivatives with MCH Antagonistic Activity and Medicaments Comprising These Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-05 US disclosed
US-20080132500-A1 Antibiotic compounds MERCK SHARP & DOHME CORP. 2008-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210283138-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL9 CA12 4778/4885CA2 4689/4885CA3 4806/4885
US-20140221334-A1 KINASE INHIBITORS MAP3K20, MAP3K1, MAP3K6 CA12 4722/4885CA2 1924/4885CA3 4419/4885
US-20100197908-A1 Pyridazine Derivatives with MCH Antagonistic Activity and Medicaments Comprising These Compounds MCHR1, MCHR2, MC5R CA12 4358/4885CA2 2268/4885CA3 4694/4885
US-20100210570-A1 LINCOMYCIN DERIVATIVES AND ANTIMICROBIAL AGENTS COMPRISING THE SAME AS ACTIVE INGREDIENT LAS1L, LCLAT1, LYPLA1 CA12 4449/4885CA2 4260/4885CA3 4757/4885
US-20170283398-A1 2-AMINOPYRIMIDINE COMPOUND AND PHARMACEUTICAL COMPOSITION AND USE THEREOF EGFR, ERBB2, IGF1R CA12 4478/4885CA2 2844/4885CA3 4605/4885
US-20080132500-A1 Antibiotic compounds NRDC, MRPL21, PEPD CA12 4680/4885CA2 4584/4885CA3 4783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.