SCHEMBL8070792

SCHEMBL8070792

NC(=O)c1ccc(N)c([N+](=O)[O-])c1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
TSHR P16473 2/20 0.50
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
ALOX15 P16050 1/20 0.47
LMNA P02545 3/20 0.46
GAA P10253 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
POLB P06746 3/20 0.42
KDM4E B2RXH2 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 2/20 0.41
USP2 O75604 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
CES1 P23141 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667585 0.90 TSHR (0.54) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL30682787 0.83 TSHR (0.43) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL3295168 0.83 TSHR (0.43) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL27832802 0.81 MEN1 (0.53) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL5576910 0.81 LMNA (0.46) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL20817271 0.79 ALDH1A1 (0.45) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL6573663 0.79 KMT2A (0.57) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL5792626 0.78 TSHR (0.48) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL27802819 0.77 POLB (0.42) KMT2ATSHRALDH1A1CYP3A4TDP1
SCHEMBL3150549 0.76 ALDH1A1 (0.74) KMT2ATSHRALDH1A1CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP claimed
EP-0700287-A1 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1996-03-13 EP claimed
WO-1994027584-A2 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1994-12-08 WO claimed